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Migration studies and toxicity evaluation of cyclic polyesters oligomers from food packaging adhesives.Sara Ubeda et al.Food chemistry, 311, 125918-125918 (2019-12-24) Androgen Receptor Signaling Reduces the Efficacy of Bacillus Calmette-Guérin Therapy for Bladder Cancer via Modulating Rab27b-Induced Exocytosis.Taichi Mizushima et al.Molecular cancer therapeutics, 19(9), 1930-1942 (2020-08-02) Suppression of mutant androgen receptors by flutamide.Junichiro Ishioka et al.International journal of urology : official journal of the Japanese Urological Association, 16(5), 516-521 (2009-04-25) The mixture effects of bisphenol derivatives on estrogen receptor and androgen receptor.Choa Park et al.Environmental pollution (Barking, Essex : 1987), 260, 114036-114036 (2020-01-30) QSAR models for anti-androgenic effect--a preliminary study.G E Jensen et al.SAR and QSAR in environmental research, 22(1-2), 35-49 (2011-03-11) Androgen receptor coregulators NOCR1, TIF2, and ARA70 may account for the hydroxyflutamide insensitivity of prostate cancer cells.Y Wang et al.Irish journal of medical science, 180(4), 865-872 (2011-07-13) Fluorescence lifetime imaging microscopy for the monitoring of green fluorescent protein-tagged androgen receptors in living cells.Rina Miyake et al.Chemical & pharmaceutical bulletin, 61(1), 82-84 (2013-01-11) Halowax 1051 affects steroidogenesis by down-regulation of aryl hydrocarbon and estrogen receptors and up-regulation of androgen receptor in porcine ovarian follicles.Justyna Barć et al.Chemosphere, 144, 467-474 (2015-09-21) Enzalutamide as an androgen receptor inhibitor prevents urothelial tumorigenesis.Takashi Kawahara et al.American journal of cancer research, 7(10), 2041-2050 (2017-11-10) Metabolism of UV-filter benzophenone-3 by rat and human liver microsomes and its effect on endocrine-disrupting activity.Yoko Watanabe et al.Toxicology and applied pharmacology, 282(2), 119-128 (2014-12-22) Determination of 2-hydroxyflutamide in human plasma by liquid chromatography-tandem mass spectrometry (LC-MS/MS): application to a bioequivalence study on Chinese volunteers.Heng Zheng et al.Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 878(19), 1611-1615 (2010-04-30) Production of human metabolites of the anti-cancer drug flutamide via biotransformation in Cunninghamella species.Jessica Amadio et al.Biotechnology letters, 33(2), 321-326 (2010-10-12) Systematic structure-function analysis of androgen receptor Leu701 mutants explains the properties of the prostate cancer mutant L701H.Dennis J van de Wijngaart et al.The Journal of biological chemistry, 285(7), 5097-5105 (2009-12-17) Development of a dual luciferase activity and fluorescamine protein assay adapted to a 384 micro-well plate format: Reducing variability in human luciferase transactivation cell lines aimed at endocrine active substances.Jennifer C Brennan et al.Toxicology in vitro : an international journal published in association with BIBRA, 47, 18-25 (2017-11-07) Anticancer Drugs That Modulate Hormone Action Medicinal Chemistry of Anticancer Drugs, 81-131 (2015) In silico binding of 4,4'-bisphenols predicts in vitro estrogenic and antiandrogenic activity.Otakuye Conroy-Ben et al.Environmental toxicology, 33(5), 569-578 (2018-02-03) A novel steroidal antiandrogen targeting wild type and mutant androgen receptors.Thomas Andrieu et al.Biochemical pharmacology, 82(11), 1651-1662 (2011-09-13) Comparing the androgenic and estrogenic properties of progestins used in contraception and hormone therapy.Renate Louw-du Toit et al.Biochemical and biophysical research communications, 491(1), 140-146 (2017-07-18) Androgen Receptor Signaling Reduces Radiosensitivity in Bladder Cancer.Hiroki Ide et al.Molecular cancer therapeutics, 17(7), 1566-1574 (2018-05-04) Effects of testosterone and 2-hydroxyflutamide on progesterone receptor expression in porcine ovarian follicles in vitro.Malgorzata Duda et al.Reproductive biology, 12(4), 333-340 (2012-12-12) Prenatal exposure to testosterone induces cardiac hypertrophy in adult female rats through enhanced Pkcδ expression in cardiac myocytes.Min Hou et al.Journal of molecular and cellular cardiology, 128, 1-10 (2019-01-15) ARHGAP15 in Human Breast Carcinoma: A Potent Tumor Suppressor Regulated by Androgens.Kiyoshi Takagi et al.International journal of molecular sciences, 19(3) (2018-03-15) Is the "comb over" dying? A mouse model for male pattern baldness (androgenic alopecia).William H Walker Endocrinology, 151(5), 1981-1983 (2010-04-23) Transport, metabolism, and hepatotoxicity of flutamide, drug-drug interaction with acetaminophen involving phase I and phase II metabolites.Seva E Kostrubsky et al.Chemical research in toxicology, 20(10), 1503-1512 (2007-09-29) Administration of flutamide alters sperm ultrastructure, sperm plasma membrane integrity and its stability, and sperm mitochondrial oxidative capability in the boar: in vivo and in vitro approach.M Lydka et al.Reproduction in domestic animals = Zuchthygiene, 47(4), 635-643 (2011-11-05) Androgens inhibit aromatase expression through DAX-1: insights into the molecular link between hormone balance and Leydig cancer development.Pamela Maris et al.Endocrinology, 156(4), 1251-1262 (2015-01-21) A mouse model of androgenetic alopecia.Judy S Crabtree et al.Endocrinology, 151(5), 2373-2380 (2010-03-18) De Facto Water Reuse: Bioassay suite approach delivers depth and breadth in endocrine active compound detectionKakaley E K, et al. The Science of the Total Environment, 699, 134297-134297 (2020) Assessment of androgen receptor agonistic/antagonistic effects on 25 chemicals in household applicants by OECD in vitro stably transfected transcriptional activation assays.Hee-Seok Lee et al.Chemosphere, 191, 589-596 (2017-10-27) A new prostate cancer therapeutic approach: combination of androgen ablation with COX-2 inhibitor.Yi Cai et al.International journal of cancer, 123(1), 195-201 (2008-04-05) ATF2 promotes urothelial cancer outgrowth via cooperation with androgen receptor signaling.Satoshi Inoue et al.Endocrine connections, 7(12), 1397-1408 (2018-12-07) Metabolomics-on-a-chip of hepatotoxicity induced by anticancer drug flutamide and Its active metabolite hydroxyflutamide using HepG2/C3a microfluidic biochips.Leila Choucha Snouber et al.Toxicological sciences : an official journal of the Society of Toxicology, 132(1), 8-20 (2012-07-31) Medroxyprogesterone acetate enhances monocyte-endothelial interaction under flow conditions by stimulating the expression of cell adhesion molecules.Fumitake Ito et al.The Journal of clinical endocrinology and metabolism, 99(6), 2188-2197 (2014-03-13) Computationally identified novel diphenyl- and phenylpyridine androgen receptor antagonist structures.Annu A Söderholm et al.Journal of chemical information and modeling, 48(9), 1882-1890 (2008-08-21) GATA3 in the urinary bladder: suppression of neoplastic transformation and down-regulation by androgens.Yi Li et al.American journal of cancer research, 4(5), 461-473 (2014-09-19) Engineered repressors are potent inhibitors of androgen receptor activity.Greg N Brooke et al.Oncotarget, 5(4), 959-969 (2014-03-25) ELK1 promotes urothelial tumorigenesis in the presence of an activated androgen receptor.Satoshi Inoue et al.American journal of cancer research, 8(11), 2325-2336 (2018-12-18) Prenatal exposure to testosterone induces cardiac hypertrophy in adult female rats through enhanced Pkc delta expression in cardiac myocytesHou M, et al. Journal of Molecular and Cellular Cardiology, 128, 1-10 (2019) Development of a novel cell based androgen screening model.Carmela Campana et al.The Journal of steroid biochemistry and molecular biology, 156, 17-22 (2015-11-20) Androgen receptors in the posterior bed nucleus of the stria terminalis increase neuropeptide expression and the stress-induced activation of the paraventricular nucleus of the hypothalamus.Brenda Bingham et al.Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 36(7), 1433-1443 (2011-03-18) Plasma glucocorticogenic activity, race/ethnicity and alcohol intake among San Francisco Bay Area women.Phum Tachachartvanich et al.PloS one, 15(6), e0233904-e0233904 (2020-06-02) TRPM8 channel as a novel molecular target in androgen-regulated prostate cancer cells.Swapna Asuthkar et al.Oncotarget, 6(19), 17221-17236 (2015-05-20) Does 2-hydroxyflutamide inhibit apoptosis in porcine granulosa cells? - An in vitro study.Malgorzata Duda et al.The Journal of reproduction and development, 58(4), 438-444 (2012-04-24) The regulation of hydroxysteroid 17β-dehydrogenase type 1 and 2 gene expression in breast cancer cell lines by estradiol, dihydrotestosterone, microRNAs, and genes related to breast cancer.Erik Hilborn et al.Oncotarget, 8(37), 62183-62194 (2017-10-06) Effects of unintentional PCBs in pigments and chemical products on transcriptional activity via aryl hydrocarbon and nuclear hormone receptors.Shinji Takeuchi et al.Environmental pollution (Barking, Essex : 1987), 227, 306-313 (2017-05-14) Androgen receptor signals regulate UDP-glucuronosyltransferases in the urinary bladder: a potential mechanism of androgen-induced bladder carcinogenesis.Koji Izumi et al.Molecular carcinogenesis, 52(2), 94-102 (2011-11-17) The synthetic progestin, gestodene, affects functional biomarkers in neonatal rat osteoblasts through an estrogen receptor-related mechanism of action.Juana Enríquez et al.Endocrine research, 42(4), 269-280 (2017-03-23) Analytical strategies to detect enobosarm administration in bovines.Nora Cesbron et al.Food additives & contaminants. Part A, Chemistry, analysis, control, exposure & risk assessment, 34(4), 632-640 (2016-11-10) Modulation of androgen receptor signaling in hormonal therapy-resistant prostate cancer cell lines.Rute B Marques et al.PloS one, 6(8), e23144-e23144 (2011-08-11) Improvement of neuronal bioenergetics by neurosteroids: implications for age-related neurodegenerative disorders.Amandine Grimm et al.Biochimica et biophysica acta, 1842(12 Pt A), 2427-2438 (2014-10-05) Nandrolone decreases mu opioid receptor expression in SH-SY5Y human neuroblastoma cells.Goffredo Guarino et al.Neuroreport, 19(11), 1131-1135 (2008-07-04) The ability of the YAS and AR CALUX assays to detect the additive effects of anti-androgenic fungicide mixtures.Bettina Seeger et al.Toxicology letters, 241, 193-199 (2015-11-26) Risk of false positive results to SARM S-4 in case of therapeutic use of antineoplastic/antiandrogen drug containing flutamide: a case study.L Perrenoud et al.Drug testing and analysis, 8(11-12), 1109-1113 (2016-08-12) Comparison of the three SARMs RAD-140, GLPG0492 and GSK-2881078 in two different in vitro bioassays, and in an in silico androgen receptor binding assay.Oliver Zierau et al.The Journal of steroid biochemistry and molecular biology, 189, 81-86 (2019-03-03) Androgen Maintains Intestinal Homeostasis by Inhibiting BMP Signaling via Intestinal Stromal Cells.Xin Yu et al.Stem cell reports, 15(4), 912-925 (2020-09-12) Testosterone inhibits matrix metalloproteinase-1 production in human endometrial stromal cells in vitro.Tomonori Ishikawa et al.Reproduction (Cambridge, England), 133(6), 1233-1239 (2007-07-20) Suppression of androgen receptor enhances the self-renewal of mesenchymal stem cells through elevated expression of EGFR.Chiung-Kuei Huang et al.Biochimica et biophysica acta, 1833(5), 1222-1234 (2013-01-22) Hydroxyflutamide enhances cellular sensitivity to 5-fluorouracil by suppressing thymidylate synthase expression in bicalutamide-resistant human prostate cancer cells.Rumi Kawabata et al.International journal of oncology, 38(3), 665-676 (2011-01-19) FOXO1 as a tumor suppressor inactivated via AR/ERβ signals in urothelial cells.Hiroki Ide et al.Endocrine-related cancer, 27(4), 231-244 (2020-02-08)

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